Gesamtpublikationsliste

2024

286   A. Horn, E. Papadopoulos, T. Kinsinger, J. Greve, E. Bickel, S. Pachoula, U. Kazmaier, "Stereoselective Synthesis of α-Azido Esters and α-Amino Acid Derivatives via Matteson Homologation of Boronic Esters", Z. anorg. allg. Chem. 2024, e202400113. DOI: 10.1002/zaac.202400113

285   Y. Hu, D. Mostert, C. Orgler, O. Andler, H. Zischka, U. Kazmaier, A. M. Vollmar, S. Braig, S. A. Sieber, S. Zahler, "Thermal Proteome Profiling Reveals Insight to Antiproliferative and Pro-Apoptotic Effects of Lagunamide A in the Modulation of DNA Damage Repair", ChemBioChem 2024, 25, e202400024. DOI: 10.1002/cbic.202400024

284   A. Siebert, U. Kazmaier, "Chemical Ligation-Mediated Total Synthesis of Corramycin", Org. Lett. 2024, 26, 3169-3173. DOI: 10.1021/acs.orglett.4c00774

283   C. Prudel, U. Kazmaier, "Total Synthesis of Moiramide B using an Allylic Alkylation Approach", Synlett 2024, in press. DOI: 10.1055/s-0042-1751578

282   M. Tost, U. Kazmaier, "Synthesis and Late-Stage Modification of (–)‑Doliculide Derivatives Using Matteson's Homologation Approach", Mar. Drugs 2024, 22, 165. DOI: 10.3390/md22040165

281   L. Junk, V. M. Schmiedel, S. Guha, K. Fischel, P. Greb, K. Schwechel, V. Krisilia, L. van Geelen, K. Rumpel, P. Kaur, R. V. Krishna­murthy, S. Narayanan, C. Kofink, A. Mantoulidis, P. Biber, G. Gmaschitz, U. Kazmaier, A. Meinhart, J. Leodolter, D. Hoi, S. Junker, F. E. Morreale, T. Clausen, R. Kalscheuer, H. Weinstabl, G. Boehmelt, "Homo-BacPROTAC-induced degradation of ClpC1 as a strategy against drug-resistant mycobacteria", Nature Commun. 2024, 15, 2005. DOI: 0.1038/s41467-024-46218-7

280   O. Andler, U. Kazmaier, "Matteson Homologation-Based Total Synthesis of Meliponamycin A", Org. Lett. 2024, 26, 148–152. DOI: 10.1021/acs.orglett.3c03766

2023

279   M. Kempf, O. Andler, U. Kazmaier, "Total synthesis of Salviachinensine A using Matteson's homologation approach", Helv. Chim. Acta 2023, e202300136. DOI: 10.1002/hlca.202300136

278   M. Tost, U. Kazmaier, "Stereoselective Synthesis of Secondary and Tertiary Boronic Esters via Matteson Homologation", Org. Lett. 2023, 25, 6835–6839. DOI: 10.1021/acs.orglett.3c02360

277  T. F. Primke, R. Ingelfinger, M. A. F. Elewa, I. Macinkovic, A. Weigert, M. P. Fabritius, C. A. Reichel, A. Ullrich, U. Kazmaier, L. D. Burgers, R. Fürst, " The Microtubule-Targeting Agent Pretubulysin Impairs the Inflammatory Response in Endothelial Cells by a JNK-Dependent Deregulation of the Histone Acetyltransferase Brd4", Cells 2023, 12, 2112. DOI: 10.3390/cells12162112

276   M. Kohr, U. Kazmaier, "Synthesis of HC-Toxin via Matteson Homologation and C-H-Functionalization", J. Org. Chem. 2023, 88, 10869–10880. DOI: 10.1021/acs.joc.3c00914

275   M. Kohr, N. Papenkordt, M. Jung, U. Kazmaier, "Total synthesis and biological evaluation of histone deacetylase inhibitor WF-3161", Org. Biomol. Chem. 2023, 21, 4382−4387. DOI: 10.1039/D3OB00641G.

274   K. Bauer, U. Kazmaier, "First Total Synthesis of Thiamyxins A-C and Thiamyxin E, a Potent Class of RNA-Virus Inhibiting (Cyclo)depsipeptides", Angew. Chem.2023, 135, 202305445. DOI: 10.1002/anie.202305445.

273   T. Kinsinger, U. Kazmaier, "Stereoselective synthesis of five- and six-membered carbocycles via Matteson homologation / ring closing metathesis", Org. Chem. Front. 2023, 10, 2963−2967. DOI: 10.1039/D3QO00457K.

272   T. Kinsinger, P. L. Schäfer, U. Kazmaier, "Stereoselective Synthesis of Highly Substituted O-Heterocycles via Matteson Homologation: a Ring-Closing Metathesis Approach", Org. Lett. 2023, 25, 3303–3307. DOI: 10.1021/acs.orglett.3c01099.

271   R. Priester, U. Kazmaier, "A Straightforward Synthesis of Emericellamide A using Matteson’s Homologation Approach", Synlett 2023, 34, 2159-2164. DOI: 10.1055/a-2077-2113.

270   D. M. Hoi, S. Junker, L. Junk, K. Fischel, D. Podlesainski, K. Schwechel, F. Kasani, L. van Geelen, J. Leodolter, P. Hawkins, F. E. Morreale, S. Kleine, S. Guha, K. Rumpel, V. M. Schmiedel, H. Weinstabl, A. Meinhart, R. Kalscheuer, R. J. Payne, M. Kaiser, M. Hartl, G. Boehmelt, U. Kazmaier, T. Clausen, "Development of a dual Clp-targeting BacPROTAC that impairs mycobacterial proteostasis and survival", Cell 2023, 186, 2176–2192. DOI: 10.1016/j.cell.2023.04.009.

2022

269   T. Kinsinger, U. Kazmaier, "Combining Matteson Homologations and Claisen Rearrange­ments - An Efficient Tool for Amino Acid Synthesis",  Eur. J. Org. Chem. 2022, e202201345. DOI: 10.1002/ejoc.202201345.

268   M. Kohr, C. Walt, J. Dastbaz, R. Müller, U. Kazmaier, "Total Synthesis of Myxoprincomid, a secondary metabolite from Myxococcus xanthus", Org. Biomol. Chem. 2022, 20, 9609–9612. DOI: 10.1039/D2OB02021A .

267   J. Greve, A. Mogk, U. Kazmaier, "Total Synthesis and Biological Evaluation of Modified Ilamycin Derivatives", Mar. Drugs 2022, 20, 632. DOI: 10.3390/md20100632.

266   A. Horn, U. Kazmaier, "Stereoselective Synthesis of the Sidechain of Callipeltin A", Org. Lett. 2022, 24, 7072–7076. DOI: 10.1021/acs.orglett.2c02586.

265   A. Horn, U. Kazmaier, "Synthesis of the Cyclic Heptapeptide Core of Callipeltin A", Org. Chem. Front. 2022, 9, 5213−5218. DOI: 10.1039/D2QO01120D.

264   T. Kinsinger, U. Kazmaier, "Matteson Homologation of Arylboronic Esters", Eur. J. Org. Chem. 2022, e202200625. DOI: 10.1002/ejoc.202200625.

263   C. Baltes, D. Thalla, U. Kazmaier, F. Lautenschläger, "Stabilizing actin inhibits single cell migration", Front. Cell Dev. Biol. 2022, 10931880. DOI: 10.3389/fcell.2022.931880.

262   F. E. Morreale, S. Kleine, J. Leodolter, S. Junker, D. M. Hoi, S. Ovchinnikov, A. Okun, J. Kley, R. Kurzbauer, L. Junk, S. Guha, D. Podlesainski, U. Kazmaier, G. Boehmelt, H. Weinstabl, K. Rumpel, V. M. Schmiedel, M. Hartl, D. Haselbach, A. Meinhart, M. Kaiser, T. Clausen, "BacPROTACs mediate targeted protein degradation in bacteria", Cell 2022, 185, 2203-2205. DOI: 10.1016/j.cell.2022.05.009.

261   T. Kinsinger, U. Kazmaier, "Application of Vinyl Nucleophiles in Matteson Homologations", Org. Lett. 2022, 24, 3599−3603. DOI: 10.1021/acs.orglett.2c01119.

260   O. Andler, U. Kazmaier, "Stereoselective Synthesis of a Protected Side Chain of Meliponamycin A", Org. Lett. 2022, 24, 2541−2545. DOI: 10.1021/acs.orglett.2c00701.

259   N. Neis, F. Xie, D. Krug, H. Zhao, A. Siebert, T. Binz, C. Fu, R. Müller, U. Kazmaier, "Stereoselective Syntheses of Deuterated Pipecolic Acids as Tools to Investigate the Stereoselectivity of the Hydroxylase GetF", Eur. J. Org. Chem. 2022, e202200162. DOI: 10.1002/ejoc.202200162.

258   V. Jakob, B. G. E. Zoller, J. Rinkes, Y. Wu, A. F. Kiefer, M. Hust, S. Helmsing, A. M. White, P. J. Harvey, T. Durek, D. J. Craik, A. Siebert, U. Kazmaier, M. Empting, "Phage Display-based Discovery of Cyclic Peptides against the Broad Spectrum Bacterial Anti-Virulence Target CsrA", Eur. J. Med. Chem. 2022, 231, 114148. DOI: 10.1016/j.ejmech.2022.114148.

257   P. Servatius, U. Kazmaier, "Synthesis and late stage modifications of Cyl-derivatives", Beilstein J. Org. Chem. 2022, 18, 174–181. DOI: 10.3762/bjoc.18.19.

2021

256   M. Tost, O. Andler, U. Kazmaier, "A Matteson homologation-based synthesis of doliculide and derivatives", Eur. J. Org. Chem. 2021, 6459–6471. DOI: 10.1002/ejoc.202101345.

255   O. Andler, U. Kazmaier, "Application of Allylzinc Reagents as Nucleophiles in Matteson Homologations", Org. Lett. 2021, 23, 8439–8444. DOI: 10.1021/acs.orglett.1c03164.

254   S. Wang, M. Meixner, L. Yu, L. Karmann, U. Kazmaier, A. M. Vollmar, I. Antes, S. Zahler, "Turning the Actin Nucleating Compound Miuraenamide into Nucleation Inhibitors", ACS Omega 2021, 6, 22165–22172. DOI: 10.1021/acsomega.1c02838.

253   L. Franz, U. Kazmaier, A. W. Truman, J. Koehnke, "Bottromycins - Biosynthesis, Synthesis and Activity", Nat. Prod. Rep. 2021, 38, 1659-1683. DOI: 10.1039/d0np00097c.

252   U. Kazmaier, L. Junk, "The Synthesis of Ilamycins/Rufomycins and Cyclomarins, Marine Cyclopeptides that Demonstrate anti-Malaria and anti-Tuberculosis Activity", Mar. Drugs 2021, 19, 446. DOI: 10.3390/md19080446.

251   M. Kohr, U. Kazmaier, "C–H Functionalization of Peptides via Cyclic Aminal Intermediates", Org. Lett. 2021, 23, 5947-5951. DOI: 10.1021/acs.orglett.1c02041.

250   O. Andler, U. Kazmaier, "Total Synthesis of Apratoxin A and B using Matteson's Homologation Approach", Org. Biomol. Chem. 2021, 19, 4866–4870. DOI: 10.1039/d1ob00713k.

249   L. Junk, E. Papadopoulos, U. Kazmaier, "Tryptophan N¹-Alkylation: Quick and Simple Access to Diversely Substituted Tryptophans", Synthesis 2021, 53, 2503–2511. DOI: 10.1055/a-1404-5079.

248   S. Kappler, U. Kazmaier, "Synthesis of modified miuraenamides – the Ugi approach", Arkivoc 2021, IV, 280–296. DOI: 10.24820/ark.5550190.p011.186.

247   S. Kappler, A. Siebert, U. Kazmaier, "Synthesis of New Cyclopeptide Analogues of the Miuraenamides", Curr. Org. Synth. 2021, 18, 418–424. DOI: 10.2174/1570179418666210113161550.

246   O. Andler, U. Kazmaier, "A Straightforward Synthesis of Polyketides via Ester Dienolate Matteson Homologation", Chem. Eur. J. 2021, 27, 949–953. DOI: 10.1002/chem.202004650.

245   U. Kazmaier, "The Long, Long Way to Bottromycin", Isr. J. Chem. 2021, 61, 302–321. DOI: 10.1002/ijch.202000068.

2020

244   L. Junk, U. Kazmaier, "The Allylic Alkylation of Ketone Enolates", ChemistryOpen 2020, 9, 929–952. DOI: 10.1002/open.202000175.

243   P. Chitirala, K. Ravichandran, C. Schirra, H.-F. Chang, E. Krause, U. Kazmaier, M. A. Lauterbach, J. Rettig, "Role of V-ATPase a3-Subunit in Mouse CTL Function", J. Immunol. 2020, DOI: 10.4049/jimmunol.1901536.

242   C. Prudel, K. Huwig, U. Kazmaier, “Stereoselective Allylic Alkylations of Amino Ketones and their Application in the Synthesis of Highly Functionalized Piperidines”, Chem. Eur. J. 2020, 26, 3181–3188, DOI: 10.1002/chem.202000051.

2019

241   I. Truebenbach, W. Zhang, Y. Wang, S. Kern, M. Höhn, S. Reinhard, J. Gorges, U. Kazmaier, E. Wagner, "Co-delivery of pretubulysin and siEG5 to EGFR 2 overexpressing carcinoma cells", Int. J. Pharm. 2019, DOI: 10.1016/j.ijpharm.2019.118570.

240   S. Wang, A. Crevenna, I. Ugur, A. Marion, I. Antes, U. Kazmaier, M. Hoyer, D. Lamb, F. Gegenfurtner, Z. Kliesmete, C. Ziegenhain, W. Enard, A. Vollmar, S. Zahler, "Actin stabilizing compounds show specific biological effects due to their binding mode", Sci. Rep. 2019, 9, 9731, DOI: 10.1038/s41598-019-46282-w.

239   A. Horn, U. Kazmaier, "Stereoselective Modification of “α-Hydroxyacid Dipeptides” by Palladium Catalyzed Allylic Alkylation", Org. Lett. 2019, 21, 4595-4599, DOI: 10.1021/acs.orglett.9b01497.

238   T. Kinsinger, U. Kazmaier, "Mono-selective β-C–H arylation of N-methylated amino acids and peptides promoted by 2-(methylthio)aniline directing group", Org. Biomol. Chem. 2019, 17, 5595-5600, DOI: 10.1039/C9OB00966C.

237   I. Truebenbach, S. Kern, D. Loy, J. Gorges, U. Kazmaier, E. Wagner, "Combination chemotherapy of L1210 tumors in mice with pretubulysin and methotrexate nanomicelles", Mol. Pharmaceut. 2019, 16, 2405-2417, DOI: 10.1021/acs.molpharmaceut.9b00038.

236   A. Kiefer, C. D. Bader, J. Held, A. Esser, J. Rybniker, M. Empting, R. Müller, U. Kazmaier, "Synthesis of New Cyclomarin Derivatives and Their Biological Evaluation towards Myco­bacterium Tuberculosis and Plasmodium Falsiparum", Chem. Eur. J. 2019, 25, 8894-8902, DOI: 10.1002/chem.201901640.

235   P. Servatius, T. Stach, U. Kazmaier, "Total synthesis of luminmycin A, a cryptic natural product from Photorhabdus luminescens", Eur. J. Org. Chem. 2019, 3163-3168, DOI: 10.1002/ejoc.201900460.

234   M. Kohr, U. Kazmaier, "Halogenated allyl alcohol derivatives – versatile dielectrophiles for palladium-catalyzed allylic alkylations", Eur. J. Org. Chem. 2019, 2843–2849, DOI: 10.1002/ejoc.201900310.

233   P. Servatius, L. Junk, U. Kazmaier, "Peptide Modifications, Versatile Tools in Peptide and Natural Product Syntheses", Synlett 2019, 30, 1289-1302, DOI: 10.1055/s-0037-1612417.

232   T. Dubich, A. Lieske, S. Santag, G. Beauclair, J. Rückert, J. Herrmann, J. Gorges, G. Bäsche, U. Kazmaier, H. Hauser, M. Stadler, T. F. Schulz, D. Wirth, "An endothelial cell line infected by Kaposi's sarcoma-associated herpes virus (KSHV) allows the investigation of Kaposi's sarcoma and the validation of novel viral inhibitors in vitro and in vivo", J. Mol. Med. 2019, 97, 311–324, DOI: 10.1007/s00109-018-01733-1.

231   S. Kern, I. Trübenbach, M. Höhn, J. Gorges, U. Kazmaier, S. Zahler, A. M. Vollmar, E. Wagner, "Combined Antitumoral Effects of Pretubulysin and Methotrexate", Pharmacol. Res. Persp. 2019, e00460, DOI: 10.1002/prp2.460.

230   L. Junk, U. Kazmaier, "Total Synthesis and Configurational Revision of Mozamide A – a Hydroxy-Brunsvicamide", J. Org. Chem. 2019, 84, 2489–2500, DOI: 10.1021/acs.joc.8b02836.

229   F. Koczian, O. Naglo, J. Vomacka, B. Vick, P. Servatius, T. Zisis, B. Hettich, U. Kazmaier, S. A. Sieber, I. Jeremias, S. Zahler, S. Braig, "Targeting the ER-Mitochondria Interface Sensitizes Leukemia Cells Towards Cytostatics", Haematologica 2018, DOI: 10.3324/haematol.2018.197368.

228   A. Kiefer, U. Kazmaier, "Syntheses of Cyclomarins – Interesting Marine Natural Products with Distinct Mode of Action towards Malaria and Tuberculosis", Synthesis 2019, 51, 107–121, DOI: 10.1055/s-0037-1610377.

227   A. Kiefer, U. Kazmaier, "Synthesis of modified β-methoxyphenylalanines via diazonium chemistry and their incorporation in desoxycyclomarin analogues", Org. Biomol. Chem. 2019, 17, 88–102, DOI: 10.1039/C8Ob02777C.

2018

226   T. Kinsinger, U. Kazmaier, "C-H-Functionalization of N-Methylated Amino Acids and Peptides as Tool in Natural Product Synthesis – Synthesis of Abyssenine A and Mucronine E", Org. Lett. 2018, 20, 7726–7730.

225   S. Kappler, L. Karmann, C. Prudel, J. Herrmann, G. Caddeu, R. Müller, A. M. Vollmar, S. Zahler, U. Kazmaier, "Synthesis and biological evaluation of (modified) miuraenamides", Eur. J. Org. Chem. 2018, 6952–6965.

224   F. A. Gegenfurtner, T. Zisis, N. Al Danaf, W. Schrimpf, Z. Kliesmete, C. Ziegenhain, W. Enard, U. Kazmaier, D. C. Lamb, A. M. Vollmar, S. Zahler, "Transcriptional effects of actin binding compounds: the cytoplasm sets the tone", Cell. Mol. Life Sci. 2018, 75, 4539–4555.

223   J. Gorges, L. Kjaerulff, F. Panter, T. Hoffmann, U. Kazmaier, R. Müller, "Structure, total synthesis and biosynthesis of Chloromyxamides – myxobacterial tetrapeptides featuring an uncommon 6-chloromethyl-5-methoxypipecolic acid building block", Angew. Chem. 2018, 130, 14466–14471; Angew. Chem. Int. Ed. 2018, 57, 14270–14275.

222   P. Servatius, U. Kazmaier, "Total Synthesis of Trapoxin A, a fungal HDAC-inhibitor from Helicoma ambiens", J. Org. Chem. 2018, 83, 11341−11349.

221   L. Junk, U. Kazmaier, "Totalsynthese und Konfigurationsrevision der Keramamide A und L aus gemeinsamer Vorstufe via späte Indolsynthese", Angew. Chem. 2018, 130, 11602−11606; Angew. Chem. Int. Ed. 2018, 57, 11432−11435.

220   M. Kohr, U. Kazmaier, "Stereoselective synthesis of d₄-(S)-lysine from (S)-serine", Synthesis 2018, 50, 4690–4694.

219   P. M. Klein, S. Kern, D.-J. Lee, J. Schmaus, J. Gorges, U. Kazmaier, E. Wagner, "Folate receptor-directed orthogonal click-functionalization of siRNA lipopolyplexes for tumor cell killing in vivo", Biomaterials 2018, 178, 630−642.

218   K. Weinhäupl, J. Lelievre, A. Goldberg, U. Kazmaier, P. Schanda, H. Fraga, "The natural antibiotic Cyclomarin blocks Arginine-Phosphate induced dynamics in ClpC1 N-terminal domain – A possible mechanism of drug action", J. Biol. Chem. 2018, 293, 8379−8393.

217   J. Gorges, U. Kazmaier, "Matteson Homologation-based Total Synthesis of Lagunamide A", Org. Lett.  2018, 20, 2033−2036.

216   P. Servatius, U. Kazmaier, "Total synthesis of the natural HDAC inhibitor Cyl-1", Org. Biomol. Chem. 2018, 16, 3464–3472.

215   A. Horn, U. Kazmaier, "Purified mCPBA, a useful reagent for the oxidation of aldehydes", Eur. J. Org. Chem. 2018, 2531–2536.

2017

214   C. Moser, D. Rüdiger, F. Förster, J. von Blume, P. Yu, B. Küster, U. Kazmaier, A. M. Vollmar, S. Zahler, "Persistent inhibition of cell migration by sub-toxic doses of miuraenamide, an actin nucleator", Sci. Rep. 2017, 7, 16407; DOI: 10.1038/s41598-017-16759-7.

213   R. Schwenk, T. Stehning, I. Bischoff, A. Ullrich, U. Kazmaier, R. Fürst, "The anti-metastatic action of the microtubule-targeting agent pretubulysin is associated with the trapping of tumor cells to the endothelium", Oncotarget 2017, 77622-77633.

212   U. Kazmaier, T. Doroshenko, K. Bauer, I. Filbrich, A. Grueter, G. Jung, A. Ullrich, "Coumaryl triflates, versatile building blocks for the modification of coumarins and for fluorescence labelling", Synthesis 2017, 49, 2743-2748.

211   I. Trübenbach, J. Gorges, J. Kuhn, E. Baratti, U. Kazmaier, E. Wagner, U. Lächelt, "Sequence-Defined Oligoamide Drug Conjugates of Pretubulysin and Methotrexate for Folate Receptor Targeted Cancer Therapy", Macromol. Biosci. 2017, DOI: 10.1002/mabi.201600520.

2016

210   B. Mondal, B. Roy, U. Kazmaier, "Stereoselective Peptide Modifications via b-C(sp³)-H Arylations", J. Org. Chem. 2016, 81, 11646-11655.

209   U. Kazmaier, "Non-stabilized enolates - versatile nucleophiles in transition-metal-catalysed allylic alkylations", Org. Chem. Front. 2016, 3, 1541-1560.

208   L. Schmidt, T. Doroshenko, P. Barbie, A. Grueter, G. Jung, U. Kazmaier, "Synthesis of fluorogenic amino acids via Pd-catalyzed allylic alkylations", Synthesis 2016, 3077-3086.

207   P. Barbie, U. Kazmaier, "Total synthesis of desoxycyclomarin C and the cyclomarazines A and B", Org. Biomol. Chem. 2016, 14, 6055−6064.

206   P. Barbie, U. Kazmaier, "Total synthesis of cyclomarins A, C and D, marine cyclopeptides with interesting anti tuberculosis and anti malaria activitites", Org. Biomol. Chem. 2016, 14, 6036−6054.

205   C. K Maurer, M. Fruth, M. Empting, O. Avrutina, J. Hoßmann, S. Nadmid, J. Gorges, J. Herrmann, U. Kazmaier, P. Dersch, R. Müller, R. W Hartmann, "Discovery of the first small molecule CsrA-RNA interaction inhibitors using biophysical screening technologies", Future Med. Chem. 2016, 8, 931-947.

204   L. Junk, U. Kazmaier, "A straightforward protocol for the synthesis of functionalized tryptophan peptides via Stille coupling, azidation and photoinduced nitrene insertion", Synlett 2016, 1531-1536.

203   L. Junk, U. Kazmaier, "Synthesis of Indoles and Tryptophan Derivatives via Photoinduced Nitrene C-H Insertion", Org. Biomol. Chem. 2016, 14, 2916−2923.

202   P. Barbie, U. Kazmaier, "Total Synthesis of Cyclomarin A, a Marine Cycloheptapeptide with anti-Tuberculosis and anti-Malaria Activity", Org. Lett. 2016, 18, 204−207.

2015

201   J. Gorges, U. Kazmaier, "BEt₃-initiated thiol-en-click reactions as a versatile tool to modify sensitive substrates", Eur. J. Org. Chem. 2015, 8011–8017.

200   P. Barbie, U. Kazmaier, "Synthesis of fully protected, reverse N-prenylated (2S,3R)-3-hydroxytryptophan, a unique building block of the cyclomarins", Org. Biomol. Chem. 2015, 13, 9267–9275.

199   A. Kiefer, D. Gawas, U. Kazmaier, "A flexible Route towards α-Hydroxyesters via Pd-catalyzed allylic alkylations", Eur. J. Org. Chem. 2015, 5810–5816.

198   P. Servatius, U. Kazmaier, "A straightforward approach towards functionalized amino acids and pipecolinic acids via Ru-catalyzed allylic alkylation", Synlett 2015, 26, 2001–2005.

197   K. Huwig, K. Schultz, U. Kazmaier, "Regio- und stereoselektive Modifizierung chiraler α-Aminoketone durch Pd-katalysierte allylische Alkylierung", Angew. Chem. 2015, 127, 9248–9251; Angew. Chem. Int. Ed. 2015, 54, 9120–9123.

196   D. Becker, U. Kazmaier, "Synthesis and biological evaluation of new dichlorinated chondramide derivatives", Eur. J. Org. Chem. 2015, 4198-4213.

195   J. Hoffmann, U. Kazmaier, "Development of a new photolabile protecting group suitable for cyclizations via ring closing metathesis", Curr. Org. Synth. 2015, 12, 475-483.

194   J. Hoffmann, J. Gorges, L. Junk, U. Kazmaier, "Synthesis of Pretubulysin-Derivatives via the TubUgi-Approach", Org. Biomol. Chem. 2015, 13, 6010-6020.

193   D. Becker, U. Kazmaier, "Synthesis of Simplified Halogenated Chondramide Derivatives as new Actin-binding Agents", Eur. J. Org. Chem. 2015, 2541–2748.

192   L. Karmann, K. Schulz, J. Herrmann, R. Müller, U. Kazmaier, "Totalsynthese und biologische Evaluierung von Miuraenamiden", Angew. Chem. 2015, 127, 4585–4590; Angew. Chem. Int. Ed. 2015, 127, 4502–4507.

191   D. S. Zurabishvili, T. J. Bukia, M. O. Lomidze, M. V. Trapaidze, E. N. Elizbarashvili, S. A. Samsoniya, T. V. Doroshenko, U. Kazmaier, Chem. Heterocycl. Comp. 2015, 51, 139–145.

190   Y. Tang, S. Frewert, K. Harmrolfs, J. Herrmann, L. Karmann, U. Kazmaier, L. Xia, Y. Zhang, R. Müller, "Heterologous expression of an orphan NRPS gene cluster from Paenibacillus larvae in E. coli revealed production of sevadicin", J. Biotechnol. 2015, 194, 122-124.

189   J. Hoffmann, U. Kazmaier, "Synthesis of Cyclic Peptides via Ring Closing Metathesis of Photolabile Protecting groups", Synthesis 2015, 47, 411-420.

2014

188   J. Eirich, S. Braig, L. Schyschka, P. Servatius, J. Hoffmann, S. Fulda, S. Zahler, U. Kazmaier, S. A. Sieber, A. M. Vollmar, "Discovery and promotion of a new class of chemosensitizer reversibly inhibiting protein disulfide isomerase", Angew. Chem. 2014, 126, 13174–13179; Angew. Chem. Int. Ed. 2014, 53, 12960–12965.

187   J. Hoffmann, U. Kazmaier, "Ein einfacher Zugang zu cyclischen, photoschaltbaren Tubulysin-Derivaten", Angew. Chem. 2014, 126, 11538–11542; Angew. Chem. Int. Ed. 2014, 53, 11356–11360.

186   A. Bayer, U. Kazmaier, "Ruthenium-catalyzed Allylic Alkylations of Chelated Enolates using Vinyl Dioxolanon-2-ones", J. Org. Chem. 2014, 79, 8498−8504.

185   A. Bayer, U. Kazmaier, "Selective Peptide Modifications via Ruthenium-catalyzed Allylic Alkylations", J. Org. Chem. 2014, 79, 8491–8497.

184   A. Bayer, U. Kazmaier, "[(p-cymene)RuCl₂]₂, an Efficient Catalyst for Highly Regioselective Allylic Alkylations of Chelated Amino Acid Ester Enolates", Chem. Eur. J. 2014, 20, 10484–10491.

183   S. Firdous, U. Kazmaier, "Syntheses of Functionalized Allylamines via Lithiated Intermediates", Eur. J. Org. Chem. 2014, 3182–3187.

182   R. Kubisch, M. von Gamm, S. Braig, A. Ullrich, J. L Burkhart, L. Colling, J. Hermann, R. Müller, U. Kazmaier, A. M. Vollmar, "Simplified pretubulysin-derivatives and their  biological effects on cancer cells", J. Nat. Prod. 2014, 77, 536-542.

181   S. Thies, U. Kazmaier, "Synthesis of a-Amino-g-lactones via Pd-catalyzed intramolecular allylic alkylation of sarcosine allyl amides", Eur. J. Org. Chem. 2014, 1695-1707.

180   R. Chaudhuri, U. Kazmaier, "Stereoselective Formation of (E)-β-Alkoxy Acrylates from Fischer Carbene Complexes and Chelated Amino Acid Ester Enolates", Synlett 2014, 25, 693-695.

179   S. Braig, R. M. Wiedmann, J. Liebl, M. Singer, R. Kubisch, L. Schreiner, B. A. Abhari, E. Wagner, U. Kazmaier, S. Fulda, A. M. Vollmar, "Pretubulysin – a new option for the treatment of metastatic cancer", Cell Death Disease 2014, 5, e1001.

178   V. K. Kretzschmann, D. Gellrich, A. Ullrich, S. Zahler, A. M. Vollmar, U. Kazmaier, R. Fürst, "The novel tubulin antagonist pretubulysin exhibits profound tumor vessel disrupting properties in vitro and in vivo", Arterioscl. Thromb. Vasc. Biol. 2014, 34, 294–303.

2013

177   P. Maity, M. Klos, U. Kazmaier, "Syntheses of α-stannylated and α-iodinated enamides via molybdenum-catalyzed hydrostannation", Org. Lett. 2013, 15, 6246-6249.

176   U. Kazmaier, A. Ullrich, J. Hoffmann, "Synthetic Approaches towards Tubulysins and their Derivatives", Open Nat. Prod. J. 2013, 6, 12-30.

175   R. Chaudhuri, U. Kazmaier, "Synthesis of 2,3-Disubstituted Pyrrols Initiated by 1,4-Addition of Chelated Enolates onto Alkynyl Carbene Complexes", Organometalllics 2013, 32, 5546-5550.

174   L. Karmann, U. Kazmaier, "Thiol-Ene Click Reactions – Versatile Tools for the Modification of Unsaturated Amino Acids and Peptides", Eur. J. Org. Chem. 2013, 7101-7109.

173   J. Gorges, A. Ullrich, U. Kazmaier, "A Straightforward Approach towards Ferrocenyl Amino Acids and Peptides via Allylic Alkylation", Eur. J. Org. Chem. 2013, 4372-4378.

172   U. Kazmaier, A. Bayer, J. Deska, "Palladium-catalyzed Allylic Alkylations as Versatile Tool in Amino Acid and Peptide Modifications", Synthesis 2013, 45, 1462-1468.

171   F. Maurer, U. Kazmaier, "Isolation of an s-alkyl iridium hydride complex, formed in the (semi)hydrogenation of an β-enamidoketone", J. Org. Chem. 2013, 78, 3425-3428.

170   M. Klos, U. Kazmaier, "A Catalyst-Economic One-Pot Protocol for the Synthesis and Conversion of Functionalized Vinylstannanes", Eur. J. Org. Chem. 2013, 1726-1731.

169   D. Becker, U. Kazmaier, "The Ireland-Claisen rearrangement as a key step in the synthesis of tubuphenylalanines", J. Org. Chem. 2013, 78, 59-65.

2012

168   P. Barbie, L. Huo, R. Müller, U. Kazmaier, "Stereoselective Synthesis of Deuterium-labeld (2S)-Cyclohexenylalanine, a Biosynthetic Intermediate of the Cinnabaramides", Org. Lett. 2012, 14, 6064-6067.

167   S. Ackermann, H.-G. Lerchen, D. Häbich, A. Ullrich, U. Kazmaier, "Synthetic studies towards Bottromycin", Beilstein J. Org. Chem. 2012, 8, 1652-1656.

166   S. Datta, A. Bayer, U. Kazmaier, "Highly Stereoselective Modifications of Peptides via Pd-catalyzed Allylic Alkylation of Internal Peptide Amide Enolates", Org. Biomol. Chem. 2012, 10, 8268-8275.

165   S. Rath, J. Liebl, R. Fürst, A. Ullrich, J. L. Burkhart, U. Kazmaier, J. Herrmann, R. Müller, M. Günther, L. Schreiner, E. Wagner, A. M. Vollmar, S. Zahler, "Anti-angiogenic effects of the tubulysin precursor pretubulysin and of simplified pretubulysin derivatives", Brit. J. Pharmacol. 2012, 167, 1048-1061.

164   J. Eirich, J. L. Burkhart, A. Ullrich, A. Vollmar, S. Zahler, U. Kazmaier, S. A. Sieber, "Pretubulysin derived probes as novel tools for monitoring the microtubule network via activity-based protein profiling and fluorescence microscopy", Mol. BioSyst. 2012, 8, 2067-2075.

163   J. Herrmann, R. M. Wiedmann, Y. A. Elnakady, A. Ullrich, M. Rohde, U. Kazmaier, A. M. Vollmar, R. Müller, "Pretubulysins: from a hypothetical biosynthetic intermediate to potential lead in tumor therapie", PLoS One 2012, 7, e37416, 1-12.

162   L. Yin, S. Lucas, F. Maurer, U. Kazmaier, Q. Hu, R. W. Hartmann, "Novel Imidazol-1-ylmethyl Substituted 1,2,5,6-Tetrahydro-pyrrolo[3,2,1-ij]quinolin-4-ones as Potent and Selective CYP11B1 Inhibitors for the Treatment of Cushing’s Syndrome", J. Med. Chem. 2012, 55, 6629-6633.

161   F. Maurer, V. Huch, A. Ullrich, U. Kazmaier, "Development of catalysts for the stereoselective hydrogenation of α,β-unsaturated ketones", J. Org. Chem. 2012, 77, 5139-5143.

160   L. Wirtz, D. Auerbach, G. Jung, U. Kazmaier, "Fluorescence Labeling of Amino Acids and Peptides with 7-Aminocoumarins", Synthesis 2012, 44, 2005-2012.

159   J. L. Burkhart, U. Kazmaier, "A Click Approach towards Tubulysin-Analogues and Tubulysin-Dolastatin Chimera", RSC Advances 2012, 3785-3790.

158   K. Schultz, L. Stief, U. Kazmaier, "A Straightforward Approach towards α-Amino-β-keto esters via Acylation of Chelates Amino Acid Ester Enolates", Synthesis 2012, 600-604.

157   J. L. Burkhart, B. Diehl, M. J. Schmitt, U. Kazmaier, "A straightforward approach towards MMP-2 and MMP-9 inhibitors based on chelate Claisen rearrangements", Eur. J. Org. Chem. 2012, 567-576.

2011

156   S. Samsonia, M. V. Trapaidze, N. N. Nikoleushvili, K. G. Japaridze, J. P. Maisuradze, U. Kazmaier, "New condensed Indoline bis-spiropyrans", Chem. Heterocycl. Comp. 2011, 47, 1098-1104.

155   J. L. Burkhart, U. Kazmaier, "A straightforward approach towards protected (S)-dolaphenine (Doe), the unusual amino acid of dolastatin 10", Synthesis 2011, 4033-4036.

154   B. Diehl, T. M. Hoffmann, N. C. Müller, J. L. Burkhart, U. Kazmaier, M. J. Schmitt, "A novel yeast bioassay for high-throughput screening of matrix metalloproteinase inhibitors", Appl. Environ. Microbiol. 2011, 8573-8577.

153   L. Wirtz, U. Kazmaier, "A mild titanium-catalyzed synthesis of functionalized amino coumarines as fluorescence labels", Eur. J. Org. Chem. 2011, 7062-7065.

152   A. F. Zahoor, S. Thies, U. Kazmaier, "A straightforward approach towards combined a-amino- and a-hydroxy acids based on Passerini reactions", Beilstein J. Org. Chem. 2011, 7, 1299-1303.

151   A. F. Zahoor, U. Kazmaier, "A Straightforward Approach towards Functionalized γ-Hydroxy and Heterocyclic Amino Acids", Synthesis 2011, 3020-3026.

150   J. Deska, S. Hähn, U. Kazmaier, "Stereoselective synthesis of deuterated β-cyclohexenyl­serine, a biosynthetic intermediate of the salinosporamides", Org. Lett. 2011, 13, 3210-3213.

149   S. Hähn, U. Kazmaier, "Chemoselective Rh-Catalyzed Allylic Alkylations of Chelated Enolates using Dienylcarbonates", Eur. J. Org. Chem. 2011, 4931-4939.

148   L. Wirtz, U. Kazmaier, "A Straightforward Approach towards Isoxazoline Amino Acids via Domino Michael Addition / Nitrile Oxide Cycloaddition", Eur. J. Org. Chem. 2011, 3467-3474.

147   J. L. Burkhart, R. Müller, U. Kazmaier, "Syntheses and Evaluation of Simplified Pretubulysin Analogues", Eur. J. Org. Chem. 2011, 3050-3059.

146   C. Bukovec, U. Kazmaier, "Stannylated allyl carbonates as versatile building blocks for the diversity oriented synthesis of allylic amines and amides", Org. Biomol. Chem. 2011, 9, 2743-2750.

145   D. Pistorius, A. Ullrich, S. Lucas, R. W. Hartmann, U. Kazmaier, R. Müller, "Biosynthesis of 2-alkyl-4(1H)-quinolones in Pseudomonas auruginosa: Potential for interference with pathogenicity", ChemBioChem 2011, 850-853.

144   A. F. Zahoor, U. Kazmaier, "A Straightforward Approach towards β-Substituted Phenyl­alanines via Ring Opening of Aryl Epoxides", Synthesis 2011, 1059-1066.

143   C. Bukovec, A. O. Wesquet, U. Kazmaier, "Insights into the Reaction Behaviour of Stannylated Allylic Substrates", Eur. J. Org. Chem. 2011, 1047-1056.

142   U. Kazmaier, A. F. Zahoor, "Regioselective Ringopening of Epoxides by Chelated Amino Acid Ester Enolates", Arkivoc 2011, IV, 6-16.

141   B. V. Lakshmi, U. K. Wefelscheid, U. Kazmaier, "Synthesis of Arylstannanes from Silyl Triflates via Aryne Intermediates", Synlett 2011, 345-348.

140   S. Datta, U. Kazmaier, "Stereoselective palladium-catalyzed allylic alkylations of peptide amide enolates", Org. Biomol. Chem. 2011, 9, 872-880.

2010

139   R. Pratap, U. Kazmaier, "Synthesis of 1-Stannylated and Iodinated 1-Chloroalkenes as Versatile Synthetic Intermediates", Synlett 2010, 3073–3077.

138   U. Kazmaier, A. Persch, "A straightforward approach towards 5-substituted thiazolylpeptides via thio-Ugi-reaction", Org. Biomol. Chem. 2010, 8, 5442-5447.

137   A. Bayer, U. Kazmaier, "Highly Regioselective Ruthenium-catalyzed Allylic Alkylations of Chelated Enolates", Org. Lett. 2010, 12, 4960–4963.

136   Y. Chai, D. Pistorius, A. Ullrich, K. J. Weissman, U. Kazmaier, R. Müller, "Discovery of 23 Novel Natural Tubulysins from Angiococcus disciformis An d48 and Cystobacter SBCb004", Chem. Biol. 2010, 17, 296–309.

135   S. Samsoniya, M. Trapaidze, N. Nikoleishvili, K. Japaridze, J. Maisuradze, U. Kazmaier, "Dipyrroloquinoxaline. 1. Synthesis of a new bisspiropyrane system on the basis of benzo[e]­pyrrolo[3,2-g]-indole", Chem. Heterocycl. Comp. 2010, 1020–1022.

134   S. Samsoniya, M. Trapaidze, N. Nikoleishvili, K. Japaridze, J. Maisuradze, U. Kazmaier, "Bisindoles. 42. Synthesis of a new bisspiropyrane system on the basis of indolo[4,5-e]-indole", Chem. Heterocycl. Comp. 2010, 1016–1019.

133   A. Z. Kalatozishvili, N. L. Targamadze, I. S. Chikvaidze, S. A. Samsoniya, A. O. Wesquet, U. Kazmaier, "A Straightforward Approach towards the Synthesis of New Bis-Pyridazino-indoles", Chem. Heterocycl. Comp. 2010, 608–612.

132   S. Rachid, O. Reverman, C. Dauth, U. Kazmaier, R. Müller, "Characterization of a Novel Type of Oxidative Decarboxylase involved in the Biosynthesis of the Styryl Moiety of Chondrochloren from an acylated Tyrosine", J. Biol. Chem. 2010, 285, 12482–12489.

131   B. V. Lakshmi, U. Kazmaier, "A straightforward approach towards substituted Morita-Baylis-Hillman (MBH) products via hydrostannation of acetylenic ketones", Synlett 2010, 407-410.

130   S. Thies, U. Kazmaier, "Vinylepoxides as Versatile Substrates for Allylations of Amino Acids and Peptides", Synlett 2010, 137-141.

129   D. Gawas, U. Kazmaier, "Diastereotopos-differentiating allylic alkylation as key step in natural product synthesis", Org. Biomol. Chem. 2010, 8, 457–462.

2009

128   A. Ullrich, J. Herrmann, R. Müller, U. Kazmaier, "Synthesis and biological evaluation of pretubulysin and derivatives", Eur. J. Org. Chem. 2009, 6367-6378.

127   U. Kazmaier, C. Schmidt, "Synthesis of Furanoid Amino Acids via a Domino Michael-/ Aldol-Addition/Cyclization-Approach", Synlett 2009, 2625-2628.

126   C. Bukovec, U. Kazmaier, "A Straightforward Protocol for One-pot Allylic Aminations/Stille Couplings", Org. Lett. 2009, 11, 3518-3521.

125   U. Kazmaier, "Erdalkalimetall-katalysierte direkte Michael-, Aldol- und Mannich-Additionen", Angew. Chem. 2009, 121, 5902-5904; Angew. Chem. Int. Ed. 2009, 47, 5790-5792.

124   U. Kazmaier, C. Schmidt, "Synthesis of Highly Functionalized Proline Derivatives via a One-Pot Michael-/SN’-Addition/Cyclization-Approach", Synthesis 2009, 2435-2439.

123   A. O. Wesquet, U. Kazmaier, "Improved Protocols for Molybdenum- und Tungsten-catalyzed Hydrostannations", Adv. Synth. Catal. 2009, 1395-1404.

122   A. Ullrich, Y. Chai, D. Pistorius, Y. A. Elnakady, J. E. Herrmann, K. J. Weissman, U. Kazmaier, and R. Müller, "Pretubulysin, a potent and chemically-accessible tubulysin precursor from Angiococcus disciformis", Angew. Chem. 2009, 121, 4486-4489; Angew. Chem. Int. Ed. 2009, 47, 4422-4425.

121   M. Bauer, U. Kazmaier, "Straightforward syntheses of chiral hydroxy isocyanides", Eur. J. Org. Chem. 2009, 2360-2366.

120   C. Quirin, U. Kazmaier, "Stereoselective Synthesis of β-Branched Phenylalanine-Derivatives via Chelate-Claisen Rearrangement", Synthesis 2009, 1725-1731.

119   U. Kazmaier, C. Schmidt, "Synthesis of Highly Functionalized Proline Derivatives via a One-pot Michael-/Aldol-Addition/Cyclization-Approach", Synlett 2009, 1136-1140.

118   H. Lin, U. Kazmaier, "Molybdenum-Catalyzed α-Hydrostannations of Propargyl Amines as Key Step for the Synthesis of N-Heterocycles", Eur. J. Org. Chem. 2009, 1221-1227.

117   D. Gawas, U. Kazmaier, "Highly Diastereoselective anti-Aldol Reactions of Glycolate Titanium Enolates", J. Org. Chem. 2009, 74, 1788-1790.

116   C. Quirin, U. Kazmaier, "Synthesis of Chlamydocin via Chelate-Claisen Rearrangement", Eur. J. Org. Chem. 2009, 371-377.

115   K. Krämer, J. Deska, C. Hebach, U. Kazmaier, "A straightforward approach towards glycoamino acids and glycopeptides via Pd-catalysed allylic alkylation", Org. Biomol. Chem. 2009, 7, 103-110.

2008

114   F. Maurer, M. Bauer, S. M. Hoffmann, U. Kazmaier, "Hydroxyalkyl Thiazolines, a new Class of Highly Efficient Ligands for Carbonyl Additions", Synlett 2008, 3203-3207.

113   C. Schmidt, U. Kazmaier, "Synthesis of highly substituted pyroglutamates via a domino Michael addition / Claisen rearrangement / lactamization approach", Org. Biomol Chem. 2008, 6, 4654-4648.

112   N. S. Samsonia, A. Z. Kalatozishvili, N. L. Targamadze, I. S. Chikvaidze, S. A. Samsoniya, A. O. Wesquet, U. Kazmaier, "A Straightforward Approach towards the Synthesis of New Bis-Pyridazino-indoles", J. Heterocycl. Chem. 2008, eingereicht.

111   S. A. Samsoniya, M. Trapaidze, N. Nikoleishvili, A. O. Wesquet, U. Kazmaier, "Pyrroloindoles. Synthesis of a new spirocyclic system based on benzo[e]pyrrolo[3,2-g]indole", Chem. Heterocycl. Comp. 2008, 1260-1262.

110   D. S. Zurabishvili, M. O. Lomidze, S. A. Samosoniya, A. O. Wesquet, U. Kazmaier, "The synthesis and transformation of some 5(6)-1-adamantyl benzimidazole", Chem. Heterocycl. Comp. 2008, 44, 941-950.

109   S. Basak, U. Kazmaier, "Palladium-catalyzed Dienylations of Chelated Enolates", Eur. J. Org. Chem. 2008, 4169-4177.

108   D. Stolz, U. Kazmaier, "Rhodium-Catalyzed Allylic Alkylations as Key Steps in the Synthesis of Cyclic α-Alkylated Amino Acids", Synthesis 2008, 2288-2292.

107   N. Jena, U. Kazmaier, "Synthesis of stannylated allyl and vinyl phosphonates via molybdenum catalyzed hydrostannations", Eur. J. Org. Chem. 2008, 3852-3858.

106   N. L. Targamadze, N. S. Samsonia, D. O. Kadjrishvili, I. S. Chikvaidze, S. A. Samsoniya, A. Wesquet, U. Kazmaier, "Some new transformations of pyrroloindole. Synthesis of new derivatives of 1H,6H-pyrrolo[2,3-]indole", Proceedings of the Georgian National Academy of Sciences 2008, 34, 35-39.

105   J. Deska, U. Kazmaier, "Peptide backbone modifications", Curr. Org. Chem. 2008, 355-385.

104   A. O. Wesquet, U. Kazmaier, "Distannylierung und Silastannylierung in situ generierter Allene", Angew. Chem. 2008, 120, 3092-3096; Angew. Chem. Int. Ed. 2008, 47, 3050-3053.

103   S. Basak, U. Kazmaier, "Allylations of Chelated Enolates using Dienyl Substrates", Org. Lett. 2008, 10, 501-504.

102   C. Schmidt, U. Kazmaier, "Efficient Stereoselective Syntheses of Constrained Glutamates via Michael Induced Ring Closing Reactions", Eur. J. Org. Chem. 2008, 887-894.

101   U. Kazmaier, D. Stolz, K. Krämer, F. Zumpe, "Influences on the Regioselectivity of Palladium-catalyzed Allylic Alkylations", Chem. Eur. J. 2008, 14, 1322-1329.

2007

100   U. Kazmaier, S. Hähn, T. D. Weiss, W. F. Maier, R. Kautenburger, "Palladium-doped Mixed Oxides as "Slow Release" Catalysts for Suzuki Couplings", Synlett 2007, 2579-2583.

99   J. Deska, U. Kazmaier, "Highly Stereoselective Peptide Modifications via Palladium Catalyzed Allylic Alkylations of Chelated Peptide Enolates", Chem. Eur. J. 2007, 13, 6204-6211.

98   J. Deska, U. Kazmaier, "Stereoselektive Synthese und Umsetzung stannylierter Peptide", Angew. Chem. 2007, 119, 4654-4657; Angew. Chem. Int. Ed. 2007, 46, 4570-4573.

97   H. Lin, U. Kazmaier, "Regioselective Mo-catalyzed hydrostannations as key steps in the synthesis of functionalized amino alcohols and heterocycles", Eur. J. Org. Chem. 2007, 2839-2843.

96   U. Kazmaier, S. Dörrenbächer, A. Wesquet, S. Lucas, M. Kummeter, "Molybdenum-catalyzed Synthesis of Stannylated Allylic Alcohol Derivatives and their Synthetic Applications", Synthesis 2007, 320-326.

2006

95   D. Stolz, U. Kazmaier, R. Pick, "Aromatic Nitro Groups and their Reactions with Chelated Ester Enolates", Synthesis 2006, 3341-3347.

94   U. Kazmaier, K. Krämer, "Isomerisierungsfreie Allylische Alkylierungen via terminale π-Allyl-Palladium-Komplexe", J. Org. Chem. 2006, 71, 8950-8953.

93   D. Stolz, R. Pick, U. Kazmaier, "Chelated Ester Enolates as versatile Nucleophiles for direct nucleophilic attack on aromatic nitro groups", Synlett 2006, 1616-1618.

92   U. Kazmaier, J. Deska, A. Watzke, "Stereoselektive Palladium-katalysierte Allylierung von Peptiden", Angew. Chem. 2006, 118, 4973-4976; Angew. Chem. Int. Ed. 2006, 45, 4855-4858.

91   U. Kazmaier, D. Stolz, "Regio- und stereoselektive Rhodium-katalysierte Allylische Alkylierungen chelatisierter Enolate", Angew. Chem. 2006, 118, 3143-3146; Angew. Chem. Int. Ed. 2006, 45, 3072-3075.

90   A. O. Wesquet, S. Dörrenbächer , U. Kazmaier, "Improved protocols for the molybdenum catalyzed hydrostannations of alkynes", Synlett 2006, 1105-1109.

89   U. Kazmaier, S. Lucas, M. Klein, "Syntheses and synthetic applications of stannylated allylic alcohols", J. Org. Chem. 2006, 71, 2429-2433.

88   U. Kazmaier, M. Bauer, "A new, modular approach towards 2-(1-hydroxyalkyl)­oxazolines, effective bidentate chiral ligands", J. Organomet. Chem. 2006, 691, 2155-2158.

87   S. Dörrenbächer, U. Kazmaier, S. Ruf, "A Straightforward Approach towards Piperidines via Stille Coupling and subsequent 1,4-Addition of Amines", Synlett 2006, 547-550.

86   S. Lucas, U. Kazmaier, "Allenyl ketones as versatile Michael acceptors for the addition of chelated enolates", Synlett 2006, 255-258.

2005

85   T. Lindner, U. Kazmaier, "Substrate controlled palladium catalyzed allylic alkylations of chelated enolates – scope and limitations", Adv. Synth. Catal. 2005, 1687-1695.

84   M. Bauer, U. Kazmaier, "Synthesis of g,d-unsaturated amino acids via palladium-catalyzed allylic alkylation of chelated glycine ester enolates", Recent Res. Devel. in Organic Chem. 2005, 9, 49-69.

83   U. Kazmaier, S. Ackermann, "A straightforward approach towards thiazoles and endothiopeptides via Ugi reaction", Org. Biomol. Chem. 2005, 3, 3184-3187.

82   B. Mendler, U. Kazmaier, V. Huch, M. Veith, "A straightforward approach to iminoxazines and azetidinimines via 1,4-additions of chelated enolates towards nitroalkenes", Org. Lett. 2005, 7, 2643-2646.

81   B. Mendler, U. Kazmaier, "Diastereoselective Michael Additions of Chelated Enolate towards Nitroalkenes", Synthesis 2005, 2239-2245.

80   U. Kazmaier, A. Wesquet, "Stannylated allylsulfones as versatile new building blocks", Synlett 2005, 1271-1274.

79   B. Mendler, U. Kazmaier, "Highly Stereoselective Additions of Tin Enolates to Nitroalkenes and their Subsequent Conversion into Nitriles", Org. Lett. 2005, 7, 1715-1718.

78   U. Kazmaier, T. Lindner, "Effizienter 1,5-Chiralitätstransfer bei Palladium-katalysierten allylischen Alkylierungen chelatisierter Aminosäureesterenolate", Angew. Chem. 2005, 117, 3368-3371; Angew. Chem. Int. Ed. 2005, 44, 3303-3306.

77   R. Pick, M. Bauer, U. Kazmaier, C. Hebach, "Ammonia in Ugi Reactions - four-component versus six-component couplings", Synlett 2005, 757-760.

76   U. Kazmaier, "Aminosäuren - wertvolle Organokatalysatoren für die Synthese von Kohlenhydraten, Angew. Chem. 2005, 117, 2224-2226; Angew. Chem. Int. Ed. 2005, 44, 2186-2188.

75   U. Kazmaier, M. Klein, "Molybdenum-Catalyzed Hydrostannations of Allenoles", Chem. Commun. 2005, 501-503.

74   U. Kazmaier, C. Hebach, A. Watzke, S. Maier, H. Mues, V. Huch, "A Straightforward Approach towards Cyclic Peptides via Ring Closing Metathesis – Scope and Limitations", Org. Biomol. Chem. 2005, 3, 136-145.

2004

73   U. Kazmaier, S. Ackermann, "An improved protocol towards the synthesis of allylated isonitriles", Synlett 2004, 2576-2578.

72   M. Pohlman, U. Kazmaier, T. Lindner, "Allylic Alkylation versus Michael induced Ring Closure – Chelated Enolates as versatile Nucleophiles", J. Org. Chem. 2004, 69, 6909-6912.

71   S. Braune, M. Pohlman, U. Kazmaier, "Molybdenum-catalyzed Stannylations as Key Steps in Heterocyclic Synthesis", J. Org. Chem. 2004, 69, 468-474.

70   U. Kazmaier, M. Pohlman, "Regioselective palladium catalyzed allylic alkylations via anti/syn-π-allyl intermediates", Synlett 2004, 623-626.

69   U. Kazmaier, "Nonstabilized Enolates as Nucleophiles in Palladium Catalyzed Allylic Alkylations", Ind. J. Org. Chem. 2003, 80, Nov. 1-11.

2003

68   U. Kazmaier, C. Hebach, "Peptide Syntheses via Ugi Reactions with Ammonia", Synlett 2003, 1591-1594.

67   M. Kummeter, U. Kazmaier, "Synthesis of Monocyclic and Bicyclic Iminosugars", Eur. J. Org. Chem. 2003, 3330-3334.

66   M. Kummeter, U. Kazmaier, "Synthesis of Polyhydroxylated Amino-Cyclopentanes", Eur. J. Org. Chem. 2003, 3325-3329.

65   M. Pohlman, U. Kazmaier, "Efficient Stereoselective Syntheses of Cyclic Amino Acids via Michael Induced Ring Closing Reactions", Org. Lett. 2003, 5, 2631-2633.

64   U. Kazmaier, "Palladium Catalyzed Allylic Alkylations of Nonstabilized Enolates", Current Org. Chem. 2003, 317-328.

63   C. Hebach, U. Kazmaier, "Via Ugi-Reaction to conformational fixed cyclic peptides", J. Chem. Soc. Chem. Commun. 2003, 596-597.

62   S. Braune, U. Kazmaier, "Entwicklung eines neuen Katalysators zur Distannylierung von Alkinen", Angew. Chem. 2003, 115, 318-320; Angew. Chem. Int Ed. 2003, 42, 306-308.

2002

61   U. Kazmaier, S. Pähler, R. Endermann, D. Häbich, H.-P. Kroll, B. Riedl, "Straigtforward Syntheses of Furanomycin Derivatives and their Biological Evaluation", Bioorg. Med. Chem. 2002, 10, 3905-3913.

60   T. D. Weiß, G. Helmchen, U. Kazmaier, "Synthesis of amino acid derivatives via enantio- and diastereoselective Pd-catalyzed allylic substitutions with a non-stabilized enolate as nucleophile", J. Chem. Soc. Chem. Commun. 2002, 1270-1271.

59   U. Kazmaier, H. Mues, A. Krebs, "Asymmetric Chelated Claisen Rearrangements in the presence of chiral ligands – Scope and limitations", Chem. Eur. J. 2002, 8, 1850-1855.

58   S. Braune, U. Kazmaier, "Regioselective hydrostannations catalyzed by molybdenum isonitrile complexes", J. Organomet. Chem. 2002, 641, 26-29.

2001

57   U. Kazmaier, F. L. Zumpe, "Chelated Enolates of Amino Acid Esters – new Efficient Nucleophiles for Isomerization-free Stereoselective Palladium-Catalyzed Allylic Substitutions", Eur. J. Org. Chem. 2001, 4067-4076.

56   H. Mues, U. Kazmaier; "The Asymmetric Chelate-Claisen Rearrangement as a Key Step in the Syntheses of Non-proteinogenic Amino Acids", Synthesis 2001, 487-498.

55   R. Stürmer, B. Schäfer,V. Wolfart, H. Stahr, U. Kazmaier, G. Helmchen, "A Short and Efficient Synthesis of (S)-1-Boc-2,5-dihydro-1H-pyrrole-2-carboxylic acid", Synthesis 2001, 46-48.

54   U. Kazmaier, D. Schauß, S. Raddatz, M. Pohlman, "Preparation and Reactions of Stannylated Amino Acids", Chem. Eur. J. 2001, 7, 456-464.

2000

53   B. Goldfuss, U. Kazmaier, "Electronic Differentiations in Palladium Alkene Complexes: Trans-Phosphine Preference of Allylic Leaving Groups", Tetrahedron 2000, 56, 6493-6496.

52   H. Mues, U. Kazmaier, "A Straightforward Approach Towards Substituted cis Hydroxyprolines via Asymmetric Chelate Claisen Rearrangements", Synlett 2000, 1004-1006.

51   U. Kazmaier, M. Pohlman, D. Schauß, "Regioselective Hydrostannations Using Mo(CO)₃(CNtBu)₃ (MoBI₃) as a New, Efficient Catalyst", Eur. J. Org. Chem. 2000, 2761-2766.

50   U. Kazmaier, D. Schauß, M. Pohlman, S. Raddatz, "Application of the Molybdenum-Catalysed Hydrostannation towards a Flexible Synthesis of Substituted Unsaturated Amino Acids", Synthesis 2000, 914-917.

49   U. Kazmaier, S. Maier, F. L. Zumpe, "A Journey from Amino Acid and Peptide Chemistry to Palladium and Back", Synlett 2000, 1523-1535.

48   S. Maier, U. Kazmaier, "Modifications of Peptides via Chelate Claisen Rearrangements of Manganese Enolates", Eur. J. Org. Chem. 2000, 1241-1251.

47   U. Kazmaier, F. L. Zumpe, "Isomerisierungsfreie Palladium-katalysierte Allylierungen - Wunsch oder Wirklichkeit?", Angew. Chem. 2000, 112, 805-807; Angew. Chem. Int. Ed. Engl. 2000, 39, 802-804.

1999

46   U. Kazmaier, S. Maier, "Application of the Peptide Claisen Rearrangement towards the Synthesis of Cyclic Peptides", Org. Lett. 1999, 1, 1763-1766.

45   U. Kazmaier, "Asymmetric Syntheses of unsaturated amino acids and peptides via Chelate-Enolate Claisen Rearrangements", J. Indian. Chem. Soc. 1999, 76, Nov.-Dez. 631-639.

44   U. Kazmaier, D. Schauß, M. Pohlman, "Mo(CO)₃(CNtBu)₃, a new Efficient Catalyst for Regioselective Hydrostannations", Org. Lett. 1999, 1, 1017-1019.

43   F. L. Zumpe, U. Kazmaier, "Application of the Palladium Catalyzed N-Allylation to the Modification of Amino Acids and Peptides", Synthesis 1999, 1785-1791.

42   U. Kazmaier, "Reactions of Chelated Amino Acid Ester Enolates and Their Application to Natural Product Synthesis", Bioorganic Chemistry, Wiley-VCH, Weinheim, 1999, 201-206.

41   M. Bakke, H. Ohta, T. Sugai, U. Kazmaier, "Action of L-Aminoacylase and L-Amino Acid Oxidase on 2-Amino-3-methyl-4-pentenoic acid Stereoisomers: An Alternative Route to Stereochemically Pure Compound and the Application to the Synthesis of (R)-2-Methyl-1-butanol", Synthesis 1999, 1671-1677.

40   U. Kazmaier, F. L. Zumpe, "Chelatisierte Aminosäureesterenolate – Effiziente Nukleophile für Palladium-katalysierte Allylische Alkylierungen", Angew. Chem. 1999, 111, 1572-1574; Angew. Chem. Int. Ed. Engl. 1999, 38, 1468-1470.

39   U. Kazmaier, S. Maier, "Stereoselective Backbone Modifications of Peptides using Peptide Metal Complexes", J. Org. Chem. 1999, 64, 4574-4575.

38   U. Kazmaier, A. Krebs, "A Straightforward Synthesis of Protected Isostatine from Achiral Precursors Using the Asymmetric Chelate Claisen-Rearrangement", Tetrahedron Lett. 1999, 40, 479-482.

1998

37   P. Comba, R. Cusack, D. P. Fairlie, L. R. Gahan, G. R. Hanson, U. Kazmaier, A. Ramlow, "The Solution Structure of a Copper(II)Compound of a New Cyclic Octapeptide by EPR Spectroscopy and Force Field Calculations", Inorg. Chem. 1998, 37, 6721-6727.

36   U. Kazmaier, "Syntheses of Polyhydroxylated Piperidine Alkaloids via Reactions of Chelated Amino Acid Ester Enolates", Recent Res. Devel. in Organic Chem. 1998, 2, 351-358.

35   U. Kazmaier, S. Maier, "Application of the Chelate Enolate Claisen Rearrangement to the Modification of Peptides", J. Chem. Soc., Chem. Commun. 1998, 2535-2536.

34   F. L. Zumpe, U. Kazmaier, "A Mild Palladium Catalyzed N-Allylation of Amino Acids and Peptides", Synlett 1998, 1199-1200.

33   U. Kazmaier, R. Grandel, "A Short Synthesis of Polyhydroxylated Piperidines via Aldol Reaction of Chelated Amino Acid Ester Enolates", Eur. J. Org. Chem. 1998, 1833-1840.

32   U. Kazmaier, C. Schneider, "Application of the Asymmetric Chelate Enolate Claisen Rearrangement to the Synthesis of Unsaturated Polyhydroxylated Amino Acids", Synthesis 1998, 1321-1326.

31   C. Schneider, U. Kazmaier, "Asymmetric Syntheses of Chiral Allylic Alcohols", Synthesis 1998, 1314-1320.

30   R. Grandel, U. Kazmaier, "Short Syntheses of Polyhydroxylated α-Alkylated Amino Acids", J. Org. Chem. 1998, 63, 4524-4528.

29   C. Schneider, U. Kazmaier, "Synthesis of 5-epi-Isofagomine via Asymmetric Chelate Enolate Claisen Rearrangement", Eur. J. Org. Chem. 1998, 1155-1159.

28   F. L. Zumpe, U. Kazmaier, "Chemoselective Claisen Rearrangement of Amino Acid Esters of Enynols", Synlett 1998, 434-436.

27   U. Kazmaier, C. Schneider, "Application of the Asymmetric Chelate-Enolate Claisen Rearrangement to the Synthesis of 5-epi-Isofagomine", Tetrahedron Lett. 1998, 39, 817-818.

26   R. Grandel, U. Kazmaier, "Diastereoselective Synthesis of β-Substituted α-Methylserines via Alanine Ester Enolates", Eur. J. Org. Chem. 1998, 409-417.

25   U. Kazmaier, "A Short Synthesis of Conjugated Unsaturated Alcohols", Tetrahedron 1998, 54, 1491-1496.

1997

24   R. Grandel, U. Kazmaier, "A Short Synthesis of Azasugars via Aldol Reaction of Chelated Amino Acid Ester Enolates", Tetrahedron Lett. 1997, 38, 8009-8012.

23   U. Kazmaier, "A Short Synthesis of Conjugated Unsaturated Amides and Esters via Triphenylphosphine-catalyzed Isomerisation of Acetylenic Pentafluorphenol Esters", J. Chem. Soc., Chem. Comm. 1997, 2305-2306.

22   C. H. Görbitz, U. Kazmaier, R. Grandel, "(+/-)-tert-Butyl 3-Hydroxy-4-phenyl-2-(toluene­sulfonylamino)pentanoate-Dichloromethane (1/1): a Pseudo Centre-of-Symmetry in an Enantiomeric Pair", Acta Cryst. C 1997, 1302-1305.

21   D. Wacker, K. Weiss, U. Kazmaier, C. Wöll, "Realization of a Phenyl-Terminated Organic Surface and Its Interaction with Chromium Atoms", Langmuir 1997, 13, 6689-6696.

20   U. Kazmaier, "Application of the Chelate-Enolate Claisen Rearrangement to the Synthesis of γ,δ-Unsaturated Amino Acids", Liebigs Ann./Recueil 1997, 285-295.

1996

19   U. Kazmaier, C. H. Görbitz, "Synthesis of Allenic Amino Acids via Chelate-Controlled Ester Enolate Claisen Rearrangement", Synthesis 1996, 1489-1493.

18   A. Krebs, U. Kazmaier, "The Asymmetric Ester Enolate Claisen Rearrangement as a Suitable Method for the Synthesis of Sterically Highly Demanding Amino Acids", Tetrahedron Lett. 1996, 37, 7945-7946.

17   U. Kazmaier, C. Schneider, "Stereoselective Synthesis of Unsaturated Polyhydroxylated Amino Acids via Ester Enolate Claisen Rearrangement", Synlett 1996, 975-977.

16   U. Kazmaier, "Synthesis of Quaternary Amino Acids Containing β,γ- as well as γ,δ-Unsaturated Side Chains via Chelate-Enolate Claisen Rearrangement", Tetrahedron Lett. 1996, 37, 5351-5354.

15   U. Kazmaier, "Synthesis of γ,δ-Unsaturated Amino Acids via Ester-Enolate Claisen Rearrangement of Chelated Allylic Esters", Amino Acids 1996, 11, 283-299.

14   R. Grandel, U. Kazmaier, B. Nuber, "anti-Selective Aldol Reactions of Amino Acid Ester Enolates. Application to the Synthesis of α-Alkylated β-Hydroxyamino Acids", Liebigs Ann. 1996, 1143-1150.

13   U. Kazmaier, "Application of the Ester Enolate Claisen Rearrangement in the Synthesis of Amino Acids Containing Quaternary Carbon Centers", J. Org. Chem. 1996, 61, 3694-3699.

12   U. Kazmaier, S. Maier, "Synthesis of Sterically High Demanding α-Alkylated Amino Acids via Claisen Rearrangement of Chelated Enolates", Tetrahedron 1996, 52, 941-954.

1990-1995

11   U. Kazmaier, "Diastereoselective Synthesis of Amino Acids Containing β-Quaternary Carbon Centers via Ester-Enolate Claisen Rearrangement", Synlett 1995, 1138-1140.

10   U. Kazmaier, S. Maier, "Stereoselective Synthesis of α-Alkylated γ,δ-Unsaturated Amino Acids via Claisen Rearrangement of Chelated Enolates", J. Chem. Soc., Chem. Comm. 1995, 1991-1992.

9   U. Kazmaier, R. Grandel, "Synthesis of Sterically Demanding α-Amino-β-Hydroxy Acids via anti-Selective Aldol Reactions", Synlett 1995, 945-946.

8   U. Kazmaier, A. Krebs, "Synthese chiraler γ,δ-ungesättigter Aminosäuren durch asymmetrische Ester-Enolat-Claisen-Umlagerung", Angew. Chem. 1995, 107, 2213-2214; Angew. Chem. Int. Ed. Engl. 1995, 34, 2012-2013.

7   U. Kazmaier, A. Krebs, C. Schneider, S. Maier, R. Grandel, "Asymmetric Synthesis of γ,δ-Unsaturated Amino Acids via Ester-Enolate Claisen Rearrangement of Chelated Allylic Esters", Amino Acids 1995, 9, 69-70.

6   U. Kazmaier, "Introduction of Allylic Side Chains onto Peptides by Pd(0)-Catalyzed Ester Enolate Claisen Rearrangement", J. Org. Chem. 1994, 59, 6667-6670.

5   U. Kazmaier, "Stereoselective Synthesis of 2-(2’-Cycloalkenyl) Glycinates via [3,3] Sigmatropic Rearrangement of Chelated Ester-Enolates", Tetrahedron 1994, 50, 12895-12902.

4   U. Kazmaier, "Synthese ungesättigter Aminosäuren durch [3,3]-sigmatrope Umlagerung chelatverbrückter Glycinesterenolate", Angew. Chem. 1994, 106, 1046-1047; Angew. Chem. Int. Ed. Engl. 1994, 33, 998-999.

3   B. M. Trost, U. Kazmaier, "Internal Redox Catalyzed by Triphenylphosphin", J. Am. Chem. Soc. 1992, 114, 7933-7935.

2   U. Schmidt, A. Lieberknecht, U. Kazmaier, H. Griesser, G. Jung, J. Metzger, "Synthesis of Di- and Trihydroxyamino Acids. – Construction of lipophilic Tripalmitoyldihydroxyamino Acids", Synthesis 1991, 49-55.

1   U. Schmidt, A. Lieberknecht, U. Kazmaier, E. Haslinger, "Welche Strukturen haben Fenestin A und Fenestin B", Angew. Chem. 1990, 102, 562-563; Angew. Chem. Int. Ed. Engl. 1990, 29, 514-515.